ASP 7663

Catalog # Availability Size / Price Qty
5178/10
5178/50
ASP 7663 | CAS No. 1190217-35-6 | TRPA1 Activators
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Description: Selective TRPA1 activator

Chemical Name: (2E)-2-[7-Fluoro-1,2-dihydro-1-(2-methylpropyl)-2-oxo-3H-indol-3-ylidene]acetic acid

Purity: ≥98%

Product Details
Citations (2)
Reviews

Biological Activity

ASP 7663 is a selective TRPA1 activator (EC50 values are ~0.5 μM in human, mouse and rat). Displays little or no affinity at more than 60 other related receptors, channels and enzymes. Stimulates 5-HT release from QGP-1 cells. Exhibits an abdominal analgesic effect in vivo. Orally bioavailable.

Technical Data

M.Wt:
263.26
Formula:
C14H14FNO3
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
1190217-35-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for ASP 7663

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2 Citations: Showing 1 - 2

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