Home / Melanin-concentrating Hormone Receptor Antagonists / GW 803430

GW 803430

Catalog #: 4242 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
4242/10
4242/50
GW 803430 | CAS No. 515141-51-2 | Melanin-concentrating Hormone Receptor Antagonists
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Description: MCH1 antagonist

Chemical Name: 6-(4-Chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-thieno[3,2-d]pyrimidin-4(3H)-one

Purity: ≥95%

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Biological Activity

GW 803430 is a selective melanin-concentrating hormone receptor 1 (MCH1) antagonist (IC50 = 9.3 nM). Displays antiobesity and antidepressant-like effects in rats and mice. Orally active.

Technical Data

M.Wt:
481.99
Formula:
C25H24ClN3O3S
Solubility:
Soluble to 25 mM in 1eq. HCl
Purity:
≥95%
Storage:
Store at -20°C
CAS No:
515141-51-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold for research purposes under agreement from GlaxoSmithKline.

Product Datasheets

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