CGP 36216 hydrochloride
Chemical Name: (3-Aminopropyl)ethylphosphinic acid hydrochloride
Purity: ≥99%
Biological Activity
CGP 36216 hydrochloride is a selective GABAB antagonist. Displays activity at presynaptic receptors; ineffective at GABAB postsynaptic receptors.Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
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CGP 36216 is a selective antagonist at GABAB presynaptic receptors in rat brain.
Ong et al.
Eur.J.Pharmacol., 2001;415:191 -
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.
Froestl et al.
J.Med.Chem., 1995;38:3313
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Citation for CGP 36216 hydrochloride
The citations listed below are publications that use Tocris products. Selected citations for CGP 36216 hydrochloride include:
1 Citation: Showing 1 - 1
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Morphine disinhibits glutamatergic input to VTA DA neurons and promotes DA neuron excitation.
Authors: Chen Et al.
J Neurosci 2015;4
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