Home / Fatty Acid Amide Hydrolase (FAAH) Inhibitors / JNJ 1661010

JNJ 1661010

Catalog #: 3262
2 Citations Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
3262/10
3262/50
JNJ 1661010 | CAS No. 681136-29-8 | Fatty Acid Amide Hydrolase (FAAH) Inhibitors
1 Image
Description: Selective, reversible FAAH inhibitor

Chemical Name: N-Phenyl-4-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-piperazinecarboxamide

Purity: ≥99%

Product Details
Citations (2)
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

JNJ 1661010 is a selective, reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 = 12 nM). Brain penetrant and active in vivo.

Technical Data

M.Wt:
365.45
Formula:
C19H19N5OS
Solubility:
Soluble to 100 mM in DMSO and to 10 mM in ethanol
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
681136-29-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Thiadiazolopiperazinyl ureas as inhibitors of fatty acid amid hydrolase.
    Keith et al.
    Bioorg.Med.Chem.Lett., 2008;18:4838

Product Datasheets

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Citations for JNJ 1661010

The citations listed below are publications that use Tocris products. Selected citations for JNJ 1661010 include:

2 Citations: Showing 1 - 2

  1. The cytoprotective effects of oleoylethanolamide in Ins-Secr.g cells do not require activation of GPR119.
    Authors: Stone Et al.
    Br J Pharmacol  2012;165:2758
  2. Cannabinoid receptor-dependent and -independent anti-proliferative effects of omega-3 ethanolamides in androgen receptor-positive and -negative prostate cancer cell lines.
    Authors: Brown Et al.
    Carcinogenesis  2010;31:1584

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