Kenpaullone

Catalog # Availability Size / Price Qty
1398/10
Kenpaullone | CAS No. 142273-20-9 | Cyclin-dependent Kinase Inhibitors
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Description: GSK-3β inhibitor; also inhibits cdks

Chemical Name: 9-Bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one

Purity: ≥98%

Product Details
Citations (2)
Reviews

Biological Activity

Kenpaullone is a GSK-3beta inhibitor (IC50 = 0.23 μM). Also inhibits cyclin dependent kinases (cdks) in the sub micromolar range (reported IC50 values are 0.4, 0.68-7 and 0.85 μM for cdk1, cdk2 and cdk5, respectively). Generates induced pluripotent stem cells (iPSCs) from somatic cells when used in combination with reprogramming factors; can replace Klf4.

Technical Data

M.Wt:
327.18
Formula:
C16H11BrN2O
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at RT
CAS No:
142273-20-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for Kenpaullone

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