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ML 233

Catalog #: 5966 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
5966/10
5966/50
ML 233 | CAS No. 2080311-92-6 | Apelin Receptor Agonists
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Description: Non-peptide apelin agonist

Chemical Name: (E)-4-Methyl-5-(((phenylsulfonyl)oxy)imino)-[1,1'-bi(cyclohexane)]-3,6-dien-2-one

Purity: ≥98%

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Biological Activity

ML 233 is a non-peptide apelin receptor agonist (EC50 = 3.7 μM); exhibits >21-fold selectivity over the closely related angiotensin 1 receptor (EC50 = >79 μM).

Technical Data

M.Wt:
359.44
Formula:
C19H21NO4S
Solubility:
Soluble to 50 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2080311-92-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Apelin, Elabela/Toddler, and biased agonists as novel therapeutic agents in the cardiovascular system.
    Yang et al.
    Trends Pharmacol Sci., 2015;36:560
  2. Functional agonists of the apelin (APJ) receptor.
    Khan et al.
    Probe Reports from the NIH Molecular Libraries Program, 2011;

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