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NVS-CECR2-1

Catalog #: 5744 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
5744/10
5744/50
NVS-CECR2-1 | CAS No. 1992047-61-6 | Bromodomain Inhibitors
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Description: Potent and selective CECR2 inhibitor

Chemical Name: N-Cyclopropyl-2-(propylsulfonyl)-6-(1-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-indol-5-yl)pyrimidin-4-amine

Purity: ≥98%

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Biological Activity

NVS-CECR2-1 is a potent and selective CECR2 (cat eye syndrome chromosome region, candidate 2) inhibitor (IC50 = 47 nM). Selective for CECR2 over a panel of bromodomains.

A concentration of 1 μM is recommended for use in cellular assays.

Technical Data

M.Wt:
495.68
Formula:
C27H37N5O2S
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1992047-61-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the NVS-CECR2-1 probe summary on the SGC website.

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