Rilmenidine hemifumarate

Catalog #: 0790
1 Citation Datasheet / COA / SDS

Catalog #	Availability	Size / Price	Qty
0790/5
0790/25

Rilmenidine hemifumarate | CAS No. 207572-68-7 | Adrenergic alpha-2 Receptor Agonists

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Description: I1 ligand. Also α2 agonist

Chemical Name: 2-[N-(Dicyclopropylmethyl)amino]oxazoline hemifumarate

Purity: ≥98%

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Product Details

Citations (1)

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Biological Activity

Rilmenidine hemifumarate is an I₁-imidazoline binding site selective ligand and α₂-adrenoceptor agonist. Possesses greater I₁ vs α₂ selectivity than the prototypical compound, clonidine. Also thought to enhance autophagy; shown to increase LC3-II levels in PC12 cells.

Technical Data

M.Wt:

238.29

Formula:

C₁₀H₁₆N₂O.½C₄H₄O₄

Solubility:

Soluble to 25 mM in DMSO

Purity:

≥98%

Storage:

Store at -20°C

CAS No:

207572-68-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
Williams et al.
Nat.Chem.Biol., 2008;4:295
Rilmenidine selectivity for imidazoline receptors in human brain.
Bricca et al.
Eur.J.Pharmacol., 1989;163:373
Antiarrhythmic action of rilmenidine on adrenaline-induced arrhythmia via central imidazoline receptors in halothane-anaesthetized dogs.
Mammoto et al.
Br.J.Pharmacol., 1996;117:1744
Keeping an eye on the I site: imidazoline-preferring receptors.
Michel and Ernsberger
TIPS, 1992;13:369
Human brain imidazoline receptors: Further characterisation with [³H] clon.
Bricca et al.
Eur.J.Pharmacol., 1994;266:25

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Citation for Rilmenidine hemifumarate

The citations listed below are publications that use Tocris products. Selected citations for Rilmenidine hemifumarate include:

1 Citation: Showing 1 - 1

Activation of I(2)-imidazoline receptors enhances supraspinal mor. analgesia in mice: a model to detect agonist and antagonist activities at these receptors.
Authors: Sánchez-Blázquez Et al.
Br J Pharmacol 2000;130:146

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