SB 699551

Catalog #: 3188 Datasheet / COA / SDS

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3188/10
3188/50

SB 699551 | CAS No. 864741-95-7 | 5-HT5 Receptor Antagonists

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Description: Selective 5-ht5a antagonist

Chemical Name: N-[2-(Dimethylamino)ethyl]-N-[[4'-[[(2-phenylethyl)amino]methyl][1,1'-biphenyl]-4-yl]methyl]cyclopentanepropanamide dihydrochloride

Purity: ≥99%

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Biological Activity

SB 699551 is a selective 5-ht_5a receptor antagonist (pK_i values are 8.3, < 6.0, < 6.0, < 6.0, < 5.5 and < 5.5 for 5-ht_5a, 5-HT_1B/D, 5-HT_2A, 5-HT_2C, 5-HT_1A and 5-HT₇ receptors respectively).

Technical Data

M.Wt:

584.66

Formula:

C₃₄H₄₅N₃O.2HCl

Solubility:

Soluble to 25 mM in DMSO and to 10 mM in ethanol

Purity:

≥99%

Storage:

Store at +4°C

CAS No:

864741-95-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:

Sold for research purposes under agreement from GlaxoSmithKline

Background References

5-ht_5A receptors as a therapeutic target.
Thomas
Pharmacol.Ther., 2006;111:707
SB-69951-A (3-cyclopentyl-N-[2-(dimethylamino)ethyl]-N-[(4'-{[(2-phenylethyl)amino]methyl}-4-biphenylyl)methyl]propanamide dihydrochloride), a novel 5-ht5A receptor-selective antagonist, enhances 5-HT neuronal function: evidence for an auto
Thomas et al.
Neuropharmacology, 2006;51:566

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