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Na+ channel blocker; citrate salt of tetrodotoxin (Cat. No. 1078)
GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels
Na+ channel blocker; also I2 imidazoline ligand
Selective NaV1.8 channel blocker
Cardiac Na+ channel blocker. Antiarrhythmic
Na+ channel blocker; antiarrhythmic agent
ASIC blocker; active in vivo
Selective NaV1.7 channel blocker
NaV blocker; neuroprotective
Selective NaV1.5 channel blocker
Potent and selective NaV1.3 and NaV1.1 channel blocker
Potent and selective Nav1.7 channel blocker
Potent hNav1.4, rNav1.6 and rNav1.7 channel activator
Potent voltage-dependent NaV1.8 channel blocker
Potent and selective NaV1.8 channel blocker; active in vivo
Potent and selective Nav1.7 blocker; analgesic